Molecule Details
InChIKeyFATWEDBJJYSZOL-JUPPYLHDSA-N
Compound NameN-Hydroxy-N-[2-[4-(4-trifluoromethoxy-phenoxy)-benzenesulfonyl]-1-(2,2,5-trimethyl-[1,3]dioxolan-4-yl)-ethyl]-formamide
Canonical SMILESC[C@@H]1OC(C)(C)OC1[C@@H](CS(=O)(=O)c1ccc(Oc2ccc(OC(F)(F)F)cc2)cc1)N(O)C=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.84
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 9.0 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.7 pIC50 TTD_MultiTarget