Molecule Details
InChIKeyFAJOBNJTLWHURK-UHFFFAOYSA-N
Canonical SMILESCSc1nc(-c2ccc(F)cc2)c(-c2ccnc(Nc3ccc(NC(=S)Nc4ccc5c(c4)C(=O)OC54c5ccc(O)cc5Oc5cc(O)ccc54)cc3)c2)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB