Molecule Details
InChIKeyDZHAENXWCJQFRP-UHFFFAOYSA-N
Compound Name2-(4-Phenethyl-piperidin-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine
Canonical SMILESc1ccc(CCC2CCN(Cc3cc4ccc[nH]c-4n3)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB