Molecule Details
InChIKeyDYRUSALPYKCZDY-RYLMWKJUSA-N
Compound Name1-methyl-4-[[(2S,6R)-3-oxa-13-thiatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methyl]piperazine
Canonical SMILESCN1CCN(CC2C[C@@H]3c4ccccc4Sc4ccccc4[C@H]3O2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35367 HRH1 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB