Molecule Details
InChIKeyDYFJXOPTRKATQT-UHFFFAOYSA-N
Canonical SMILESCOc1ccc(C(=O)NCCO)cc1Nc1nccc(Oc2ccc(NC(=O)Nc3cc(C(C)C)nn3-c3ccc(C)cc3)c3ccccc23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 6.8 IC50 ChEMBL;BindingDB