Molecule Details
InChIKeyDYFDYWXRTZSUEM-UHFFFAOYSA-N
Compound Name1-(1,3-Benzothiazol-2-yl)-5-(4-pyrimidin-2-ylpiperazin-1-yl)pentan-1-one
Canonical SMILESO=C(CCCCN1CCN(c2ncccn2)CC1)c1nc2ccccc2s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P34969 HTR7 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB