Molecule Details
InChIKeyDXUMILREMTTZQK-UHFFFAOYSA-N
Compound NameUS11279703, Table 1.3
Canonical SMILESCC(C)(C)S(=O)(=O)Nc1cccc(Nc2nc(NC3CCNCC3)nc3sccc23)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 6.7 IC50 ChEMBL;BindingDB
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 6.6 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 6.3 IC50 ChEMBL;BindingDB