Molecule Details
InChIKeyDXAACKOYNNQYHC-UHFFFAOYSA-N
Compound Name2-[[5-Chloro-2-[4-(2-oxopyrrolidin-1-yl)anilino]pyrimidin-4-yl]amino]benzamide
Canonical SMILESNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCCC3=O)cc2)ncc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.68
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 9.8 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 9.6 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 9.6 IC50 ChEMBL