Molecule Details
InChIKeyDWMNINPORGJSKR-UHFFFAOYSA-N
Compound Name1-ethyl-3-[4-[1-ethyl-4-[2-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrazol-3-yl]phenyl]urea
Canonical SMILESCCNC(=O)Nc1ccc(-c2nn(CC)cc2-c2ccnc3[nH]c(-c4ccc(CN5CCOCC5)cc4)cc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.6 pIC50 TTD_MultiTarget