Molecule Details
InChIKeyDWJRVXUXEZICSB-ZDUSSCGKSA-N
Compound Name5-[3-[4-[(3S)-3-aminopiperidin-1-yl]pyrimidin-2-yl]-1H-indol-5-yl]-N-methyl-1,3,4-thiadiazol-2-amine
Canonical SMILESCNc1nnc(-c2ccc3[nH]cc(-c4nccc(N5CCC[C@H](N)C5)n4)c3c2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.1 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB