Molecule Details
InChIKeyDWHRPZRXNRDAQF-GEQJWKGNSA-N
Compound NameTyr-D-Phe-Gly-Trp-Nle-Asp-Phe-NH2
Canonical SMILESCCCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.29
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41143 OPRD1 Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P32238 CCKAR Homo sapiens Human PF00001 PF09193 7.6 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB