Molecule Details
InChIKeyDWEHMLBGRQZUJA-UHFFFAOYSA-N
Compound NameN-[4-[4-(2-methylsulfanylphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide
Canonical SMILESCSc1ccccc1N1CCN(CCCCNC(=O)c2cc3ccccn3n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB