Molecule Details
InChIKeyDVVVOLSRHWJCHV-UHFFFAOYSA-N
Compound NameN-(2,2-Difluoro-5h-[1,3]dioxolo[4,5-F]benzimidazol-6-Yl)-2-{[2-(Trifluoromethoxy)benzoyl]amino}-1,3-Thiazole-4-Carboxamide
Canonical SMILESO=C(Nc1nc2cc3c(cc2[nH]1)OC(F)(F)O3)c1csc(NC(=O)c2ccccc2OC(F)(F)F)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49674 CSNK1E Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB
Q9Y6M4 CSNK1G3 Homo sapiens Human PF12605 PF00069 6.1 IC50 ChEMBL;BindingDB