Molecule Details
InChIKeyDVTNAPPKBSPOMR-UHFFFAOYSA-N
Compound Name3-(3,4-Dichloro-phenyl)-1-(1-phenyl-2-pyrrolidin-1-yl-ethyl)-1,3,4,7-tetrahydro-azepin-2-one
Canonical SMILESO=C1C(c2ccc(Cl)c(Cl)c2)CC=CCN1C(CN1CCCC1)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 9.5 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB