Molecule Details
InChIKeyDVPJGCNYHGTCEI-QMMMGPOBSA-N
Compound Name2-[(2S)-piperidin-2-yl]-6-[5-(trifluoromethyl)-1H-pyrazol-4-yl]thieno[3,2-d]pyrimidin-4 (3H)-one
Canonical SMILESO=c1[nH]c([C@@H]2CCCCN2)nc2cc(-c3c[nH]nc3C(F)(F)F)sc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBU7 DBF4 Homo sapiens Human PF07535 9.1 IC50 ChEMBL;BindingDB
O00311 CDC7 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 6.3 IC50 ChEMBL;BindingDB