Molecule Details
InChIKeyDVOSPTOWEQEYQB-UHFFFAOYSA-N
Compound Name3-Ethyl-2-[(3-fluoro-4-pyridinyl)amino]-7-[1-(3-hydroxy-2,2-dimethylpropanoyl)piperidin-3-yl]thieno[3,2-d]pyrimidin-4-one
Canonical SMILESCCn1c(Nc2ccncc2F)nc2c(C3CCCN(C(=O)C(C)(C)CO)C3)csc2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13946 PDE7A Homo sapiens Human PF00233 8.9 IC50 ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 7.4 IC50 ChEMBL;BindingDB
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 6.7 IC50 ChEMBL;BindingDB