Molecule Details
InChIKeyDVNVXZQJDUVWTB-RWWKDMOOSA-N
Compound Name(2R)-2-[4-(2,5-dioxoimidazolidin-1-yl)cyclohexyl]-2-[[4-(4-methoxyphenyl)phenyl]sulfonylamino]acetic acid
Canonical SMILESCOc1ccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C3CCC(N4C(=O)CNC4=O)CC3)cc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.29
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.4 pIC50 TTD_MultiTarget
P45452 MMP13 Homo sapiens Human PF00045 PF00413 PF01471 7.2 IC50 ChEMBL
P18843 nadE Escherichia coli (strain K12) Pathogen PF02540 7.3 pIC50 TTD_MultiTarget