Molecule Details
InChIKeyDURNYYKOVXELMP-UHFFFAOYSA-N
Compound Name2-(2-aminoethylamino)-N-(7-methoxyquinolin-6-yl)thieno[3,2-d]pyrimidine-7-carboxamide
Canonical SMILESCOc1cc2ncccc2cc1NC(=O)c1csc2cnc(NCCN)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NWZ3 IRAK4 Homo sapiens Human PF07714 8.0 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.8 IC50 ChEMBL;BindingDB
P51617 IRAK1 Homo sapiens Human PF00531 PF00069 6.2 IC50 ChEMBL;BindingDB