Molecule Details
InChIKeyDUKZDMUZDDNVFF-UHFFFAOYSA-N
Compound Name5-[4-(3,3-dimethylpiperazin-1-yl)phenyl]-2-(7-ethyl-1H-indol-4-yl)-1,3-oxazole-4-carboxamide
Canonical SMILESCCc1ccc(-c2nc(C(N)=O)c(-c3ccc(N4CCNC(C)(C)C4)cc3)o2)c2cc[nH]c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 9.2 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB