Molecule Details
InChIKeyDUJWQCUJEVGZHQ-JOCHJYFZSA-N
Compound Name(R)-N-(4-(7-chloro-8-hydroxy-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-1-yl)benzyl)-N-cyclobutylacetamide
Canonical SMILESCC(=O)N(Cc1ccc([C@H]2CN(C)CCc3cc(Cl)c(O)cc32)cc1)C1CCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21728 DRD1 Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P21918 DRD5 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB