Molecule Details
InChIKeyDUIYQEGWIKOTCS-UHFFFAOYSA-N
Compound Name3-amino-N-[4-(2,6-diaminopyrimidin-4-yl)-3-pyridinyl]-6-(2-fluorophenyl)pyridine-2-carboxamide
Canonical SMILESNc1cc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)nc(N)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.9 Ki ChEMBL;BindingDB