Molecule Details
InChIKeyDTSANQSRTBGPPK-XMMPIXPASA-N
Compound Name(2R)-2-[(3-methoxyphenyl)carbamoylamino]-5-oxo-N,N-dipentyl-5-pyrrolidin-1-ylpentanamide
Canonical SMILESCCCCCN(CCCCC)C(=O)[C@@H](CCC(=O)N1CCCC1)NC(=O)Nc1cccc(OC)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.07
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 6.1 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB