Molecule Details
InChIKeyDTQIXKQBUYCCQM-FSEITFBQSA-N
Compound Name(2S)-N-acetyl-2-[[(2S)-2-[[(2S)-5-amino-1-oxo-1-[2-[4-[4-[1-[2-oxo-2-(6-oxo-5H-benzo[b][1,4]benzodiazepin-11-yl)ethyl]piperidin-4-yl]butyl]piperazin-1-yl]ethylamino]pentan-2-yl]amino]-4-(diaminomethylideneamino)butanoyl]amino]butanediamide
Canonical SMILESCC(=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCNC(=N)N)N[C@@H](CCCN)C(=O)NCCN1CCN(CCCCC2CCN(CC(=O)N3c4ccccc4NC(=O)c4ccccc43)CC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08172 CHRM2 Homo sapiens Human PF00001 9.8 Ki ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P08173 CHRM4 Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB