Molecule Details
InChIKeyDSWPTVKCBCROGK-QZTJIDSGSA-N
Compound NameUS9763957, Example 1
Canonical SMILESCCOC(=O)c1c(C)ccnc1O[C@@H]1CC[C@@H](C)N(C(=O)c2ccccc2-n2nccn2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43614 HCRTR2 Homo sapiens Human PF00001 PF03827 8.1 IC50 ChEMBL;BindingDB
Q13822 ENPP2 Homo sapiens Human PF01223 PF01663 PF01033 8.1 IC50 ChEMBL;BindingDB
O43613 HCRTR1 Homo sapiens Human PF00001 7.1 IC50 ChEMBL;BindingDB