Molecule Details
InChIKeyDSUYZKFAJRJFFP-UHFFFAOYSA-N
Compound Name1,4-[(Naphthalene-1,7-diyl)oxy[6-[4-(trifluoromethyl)phenyl]-1,3-phenylene]methylene(1H-imidazole-1,5-diyl)ethylene]piperazine-2-one
Canonical SMILESO=C1CN2CCc3cncn3Cc3ccc(-c4ccc(C(F)(F)F)cc4)c(c3)Oc3ccc4cccc(c4c3)N1CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.8
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P53609 PGGT1B Homo sapiens Human PF00432 7.8 IC50 ChEMBL
P49354 FNTA Homo sapiens Human PF01239 7.8 IC50 ChEMBL;BindingDB