Molecule Details
InChIKeyDSMKXMINSCXYGH-CAZXVXRPSA-N
Canonical SMILESO=C(NS(=O)(=O)c1ccc(N[C@H](CCN(CCO)CCO)CSc2ccccc2)c(S(=O)(=O)C(F)(F)F)c1)c1ccc(N2CCC([C@@H](O)c3ccccc3-c3ccc(Cl)cc3)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 9.1 IC50 ChEMBL;BindingDB
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 9.0 IC50 ChEMBL;BindingDB