Molecule Details
InChIKeyDSEZYCNDQGVNMS-SFHVURJKSA-N
Compound Name[(2S)-1-[6-[1-(6-piperazin-1-yl-2-pyridinyl)pyrazolo[4,3-c]pyridin-6-yl]pyrazin-2-yl]pyrrolidin-2-yl]methanol
Canonical SMILESOC[C@@H]1CCCN1c1cncc(-c2cc3c(cn2)cnn3-c2cccc(N3CCNCC3)n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 10.3 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 10.0 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.7 Ki ChEMBL;BindingDB