Molecule Details
InChIKeyDRRPFYALBDCXPZ-UHFFFAOYSA-N
Compound NameN-[2-[3-fluoro-4-[[4-oxo-6-(propan-2-ylcarbamoylamino)-2-propylquinazolin-3-yl]methyl]phenyl]phenyl]sulfonyl-2-(2-methylpropoxy)acetamide
Canonical SMILESCCCc1nc2ccc(NC(=O)NC(C)C)cc2c(=O)n1Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)COCC(C)C)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 8.8 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB