Molecule Details
InChIKeyDRMHBTZKBJCWJJ-UHFFFAOYSA-N
Compound Name3-amino-N-[4-(2-aminopyrimidin-4-yl)-3-pyridinyl]-6-(2,6-difluorophenyl)pyridine-2-carboxamide
Canonical SMILESNc1nccc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.3 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.2 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.3 Ki ChEMBL;BindingDB