Molecule Details
InChIKeyDRCFAJOBBUQTRU-UHFFFAOYSA-N
Compound Name4-cyano-N-[(4-cyanophenyl)methyl]-N-[(3-methylimidazol-4-yl)methyl]-5-naphthalen-1-yl-3,6-dihydro-2H-pyridine-1-carboxamide
Canonical SMILESCn1cncc1CN(Cc1ccc(C#N)cc1)C(=O)N1CCC(C#N)=C(c2cccc3ccccc23)C1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.46
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.5 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.5 IC50 ChEMBL