Molecule Details
InChIKeyDQAHFXNORWIJPU-NKQBFHEZSA-N
Compound Name(2S)-2-amino-N-[(7S,13S,18S,24S)-18-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-7,24-dibenzyl-6,9,12,19,22,25-hexaoxo-1,2,15,16-tetrathia-5,8,11,20,23,26-hexazacyclooctacos-13-yl]-3-(4-hydroxy-2,6-dimethylphenyl)propanamide
Canonical SMILESCc1cc(O)cc(C)c1C[C@H](N)C(=O)N[C@@H]1CSSC[C@@H](NC(=O)[C@@H](N)Cc2c(C)cc(O)cc2C)C(=O)NCC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCSSCCNC(=O)[C@H](Cc2ccccc2)NC(=O)CNC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 9.6 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB