Molecule Details
InChIKeyDPYNGTQCAJQNSC-UHFFFAOYSA-N
Compound Name4-[4-[[2-(4-Ethylpiperazin-1-yl)pyrimidin-4-yl]oxymethyl]triazol-1-yl]benzenesulfonamide
Canonical SMILESCCN1CCN(c2nccc(OCc3cn(-c4ccc(S(N)(=O)=O)cc4)nn3)n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 9.2 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 9.1 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 7.6 Ki ChEMBL;BindingDB