Molecule Details
InChIKeyDPSFKKBIIZTWDA-UHFFFAOYSA-N
Compound NameN-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridine-5-carboxamide
Canonical SMILESO=C(Nc1cccc(O)c1)c1cnc2[nH]cc(-c3ccc(O)cc3)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
Q9Y463 DYRK1B Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 6.1 IC50 ChEMBL;BindingDB