Molecule Details
InChIKeyDPERSSXJBGKIEL-UHFFFAOYSA-N
Compound Name1-[2-(1,4-Diazepan-1-yl)pyrimidin-4-yl]-6-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]pyrazolo[4,3-c]pyridine
Canonical SMILESFC(F)(F)Cn1cc(-c2cc3c(cn2)cnn3-c2ccnc(N3CCCNCC3)n2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.8 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.3 Ki ChEMBL;BindingDB