Molecule Details
InChIKeyDOVSNSDMRJVTMR-JOCHJYFZSA-N
Compound Name(4R)-4-(4-cyanophenyl)-N-(2-hydroxy-2-methylpropyl)-2,5-dioxo-1-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-cyclopenta[d]pyrimidine-3-carboxamide
Canonical SMILESCC(C)(O)CNC(=O)N1C(=O)N(c2cccc(C(F)(F)F)c2)C2=C(C(=O)CC2)[C@H]1c1ccc(C#N)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08246 ELANE Homo sapiens Human PF00089 9.1 IC50 ChEMBL
P24158 PRTN3 Homo sapiens Human PF00089 6.4 IC50 ChEMBL