Molecule Details
InChIKeyDOVNDOSDULTCGE-QSVHXPHUSA-N
Compound NameN-(2-(4-((3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl)piperazin-1-yl)-2-cyclohexylethyl)-N-isopropylpyridazine-3-carboxamide
Canonical SMILESCC(C)N(CC(C1CCCCC1)N1CCN(C(=O)[C@@H]2CN(C(C)(C)C)C[C@H]2c2ccc(F)cc2F)CC1)C(=O)c1cccnn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.9 IC50 ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB