Molecule Details
InChIKeyDOJSODPNZWPNBR-PPRPKMEESA-N
Compound Name(5R)-4-[(1S,6R)-5-[(2S)-2-(4-chlorophenyl)-3-(cyclopropylamino)propanoyl]-2,5-diazabicyclo[4.1.0]heptan-2-yl]-5-methyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidin-7-one
Canonical SMILESC[C@@H]1CC(=O)Nc2ncnc(N3CCN(C(=O)[C@H](CNC4CC4)c4ccc(Cl)cc4)[C@@H]4C[C@@H]43)c21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y243 AKT3 Homo sapiens Human PF00169 PF00069 PF00433 10.0 IC50 ChEMBL;BindingDB
P31749 AKT1 Homo sapiens Human PF00169 PF00069 PF00433 9.2 IC50 ChEMBL;BindingDB
P31751 AKT2 Homo sapiens Human PF00169 PF00069 PF00433 8.2 IC50 ChEMBL;BindingDB