Molecule Details
InChIKeyDOCKONDCDYZCFE-UHFFFAOYSA-N
Compound Name4-(Piperidin-4-ylamino)-6-[3-(trifluoromethoxy)anilino]-1,3,5-triazine-2-carbonitrile
Canonical SMILESN#Cc1nc(Nc2cccc(OC(F)(F)F)c2)nc(NC2CCNCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43235 CTSK Homo sapiens Human PF08246 PF00112 7.2 IC50 ChEMBL;BindingDB
P25774 CTSS Homo sapiens Human PF08246 PF00112 6.7 IC50 ChEMBL;BindingDB
P07711 CTSL Homo sapiens Human PF08246 PF00112 6.3 IC50 ChEMBL;BindingDB