Molecule Details
InChIKeyDOBIYIOPZIMMRH-AMBBWHSESA-N
Compound Name(4S)-5-[[(2S)-6-[6-[5-[(3aS,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-1-[[(2S)-1-carboxy-4-(2,6-dimethylbenzoyl)oxy-3-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-5-oxo-4-(phenylmethoxycarbonylamino)pentanoic acid
Canonical SMILESCc1cccc(C)c1C(=O)OCC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCCNC(=O)CCCCCNC(=O)CCCCC1SC[C@@H]2NC(=O)N[C@H]12)NC(=O)[C@H](CCC(=O)O)NC(=O)OCc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29466 CASP1 Homo sapiens Human PF00619 PF00656 8.2 Ki ChEMBL;BindingDB
Q14790 CASP8 Homo sapiens Human PF01335 PF00656 6.3 Ki ChEMBL;BindingDB
P42574 CASP3 Homo sapiens Human PF00656 6.1 Ki ChEMBL;BindingDB