Molecule Details
InChIKeyDNNZYGQJIKJSHH-NEEWURRISA-N
Canonical SMILESCc1cc2nc(C(C)C)[nH]c2cc1-c1ccc(C[C@H](NC(=O)[C@H]2CC[C@H](CN)CC2)C(=O)Nc2ccc(-c3nnc(C(F)(F)C(F)(F)C(=O)O)[nH]3)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 9.5 IC50 ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 9.1 IC50 ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 8.1 IC50 ChEMBL;BindingDB