Molecule Details
InChIKeyDNNYNSPBJXNYMZ-UHFFFAOYSA-N
Canonical SMILESO=C(c1ccccc1)c1cnc2c(C(F)(F)F)ccc(-c3cccc(OCc4ccc(C(Cc5ccc(-c6ccccc6)cc5)C(=O)O)cc4)c3)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P55055 NR1H2 Homo sapiens Human PF00104 PF00105 6.3 IC50 ChEMBL;BindingDB
Q13133 NR1H3 Homo sapiens Human PF00104 PF00105 6.3 IC50 ChEMBL;BindingDB