Target not found.
Molecule Details
InChIKeyDNIBTKHTGSPUNA-RHSAGAAYSA-N
Compound NameH-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys]-Thr-NH2
Canonical SMILESC[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](N)Cc2ccccc2)CSSC[C@@H](C(=O)N[C@H](C(N)=O)[C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30874 SSTR2 Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P35346 SSTR5 Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 6.3 IC50 ChEMBL;BindingDB