Molecule Details
InChIKeyDNFNQGHGGVBVSY-UHFFFAOYSA-N
Compound Name2-(dimethylamino)-1-[2-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]-7,8-dihydro-5H-1,6-naphthyridin-6-yl]-2-methylpropan-1-one
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCN(C(=O)C(C)(C)N(C)C)C5)ncc3F)cc2n1C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB