Molecule Details
InChIKeyDNDWQJKQEQLRTQ-GOGZTAQTSA-N
Compound Name(2R,4R)-1-((R)-2-((S)-2-amino-3-(1H-imidazol-4-yl)propanamido)-3-phenylpropanoyl)-N-(2-guanidinoethyl)-4-(naphthalen-2-ylmethoxy)pyrrolidine-2-carboxamide
Canonical SMILESNC(N)=NCCNC(=O)[C@H]1C[C@@H](OCc2ccc3ccccc3c2)CN1C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H](N)Cc1c[nH]cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01726 MC1R Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB