Molecule Details
InChIKeyDNCXPYGCTRGWJY-UHFFFAOYSA-N
Compound Name2-[4-[(3-Phenyltriazolo[4,5-d]pyrimidin-5-yl)amino]phenoxy]acetic acid
Canonical SMILESO=C(O)COc1ccc(Nc2ncc3nnn(-c4ccccc4)c3n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49840 GSK3A Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB