Molecule Details
InChIKeyDNASOPMPZKFRCW-UHFFFAOYSA-N
Compound Name1-(2,4-Dimethyloxazol-5-ylcarbonyl)-2,3-dihydro-8-(4-methylpiperazin-1-yl)pyrrolo[3,2-g]isoquinoline
Canonical SMILESCc1nc(C)c(C(=O)N2CCc3cc4ccnc(N5CCN(C)CC5)c4cc32)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB