Molecule Details
InChIKeyDMQMZHJLQOERFT-CQSZACIVSA-N
Compound Name4-[[[(1R)-1-carboxyethyl]-[6-[4-(diaminomethylideneamino)benzoyl]oxyquinoline-2-carbonyl]amino]methyl]thiophene-2-carboxylic acid
Canonical SMILESC[C@H](C(=O)O)N(Cc1csc(C(=O)O)c1)C(=O)c1ccc2cc(OC(=O)c3ccc(NC(=N)N)cc3)ccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07477 PRSS1 Homo sapiens Human PF00089 9.5 IC50 ChEMBL;BindingDB
P07478 PRSS2 Homo sapiens Human PF00089 9.5 IC50 ChEMBL
P35030 PRSS3 Homo sapiens Human PF00089 9.5 IC50 ChEMBL