Molecule Details
InChIKeyDMOLFVGCLPCFQX-UHFFFAOYSA-N
Compound Name4-(1-Benzylpiperidin-4-yl)-2-[(8-hydroxyquinolin-2-yl)methyl-prop-2-ynylamino]butanenitrile
Canonical SMILESC#CCN(Cc1ccc2cccc(O)c2n1)C(C#N)CCC1CCN(Cc2ccccc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P22303 ACHE Homo sapiens Human PF08674 PF00135 7.8 Ki ChEMBL;BindingDB
P06276 BCHE Homo sapiens Human PF08674 PF00135 7.3 Ki ChEMBL;BindingDB