Molecule Details
InChIKeyDMMNMIJPRNMLBQ-UHFFFAOYSA-N
Compound Name3-{3-[4-(2-Carbamoyl-phenyl)-piperazin-1-yl]-propylcarbamoyl}-4-(3,4-difluoro-phenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid methyl ester
Canonical SMILESCOC(=O)C1=C(C)NC(=O)N(C(=O)NCCCN2CCN(c3ccccc3C(N)=O)CC2)C1c1ccc(F)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.9 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB