Molecule Details
InChIKeyDMHSDGHSQKYUDC-IAGOWNOFSA-N
Compound NameUS10183947, Example 8
Canonical SMILESCn1ncc(NC(=O)[C@@H]2CCCC[C@H]2C(=O)c2ccc(-c3ccn[nH]3)cc2)c1S(C)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P09917 ALOX5 Homo sapiens Human PF00305 PF01477 7.3 IC50 ChEMBL;BindingDB
P20292 ALOX5AP Homo sapiens Human PF01124 7.3 IC50 ChEMBL
P39748 FEN1 Homo sapiens Human PF00867 PF00752 7.3 IC50 ChEMBL